Antazoline
Research News and Information

Sunday, November 22, 2009

Demand for food and cocaine in Fischer and Lewis rats.

30 Jan 2009 Fischer and Lewis rat strains often serve as animal vulnerability models for drug abuse and addiction. When these strains respond for drugs of abuse, several measures, including total drug intake, response rate and progressive-ratio breakpoints, ... Read more...

Evidence for imidazoline receptors involvement in the agmatine antidepressant-like effect in the forced swimming test.

22 Mar 2007 This study investigated the involvement of the imidazoline receptors in the antidepressant-like effect of agmatine in the forced swimming test. The antidepressant-like effects of agmatine (10 mg/kg, i.p.) in the forced swimming test was blocked by ... Read more...

A rapid derivative spectrophotometric method for simultaneous determination of naphazoline and antazoline in eye drops.

30 Dec 2005 A zero-crossing first-derivative spectrophotometric method is applied for the simultaneous determination of naphazoline hydrochloride and antazoline phosphate in eye drops. The measurements were carried out at wavelengths of 225 and 252 nm for ... Read more...

Latest indexed articles for 'Antazoline'

These are the very latest articles for this heading:

• Demand for food and cocaine in Fischer and Lewis rats. 30 Jan 2009
• Evidence for imidazoline receptors involvement in the agmatine antidepressant-like effect in the forced swimming test. 22 Mar 2007
• A rapid derivative spectrophotometric method for simultaneous determination of naphazoline and antazoline in eye drops. 30 Dec 2005
• Simple HPLC determination of benzalkonium chloride in ophthalmic formulations containing antazoline and tetrahydrozoline. 30 Aug 2005
• Influence of antazoline and ketotifen on the anticonvulsant activity of conventional antiepileptics against maximal electroshock in mice. 30 Jul 2004
• Neuroprotective activity of antazoline against neuronal damage induced by limbic status epilepticus. 30 Dec 2002
• Inhibition of voltage-gated Ca2+ channels by antazoline. 5 Oct 2002
• Effects of imidazoline binding site ligands on the growth and viability of clonal pancreatic beta-cells. 30 Jan 2000
• Protection by imidazol(ine) drugs and agmatine of glutamate-induced neurotoxicity in cultured cerebellar granule cells through blockade of NMDA receptor. 29 Jun 1999
• Influence of antazoline on the anticonvulsant activity of conventional antiepileptic drugs against maximal electroshock-induced seizures in mice. 30 Dec 1998
• Determination of antihistamines based on the formation of mixed aggregates with surfactants. 29 Apr 1998
• Antazoline increases insulin secretion and improves glucose tolerance in rats and dogs. 16 Apr 1997
• [Antazoline/tetryzoline eyedrops in comparison with levocabastine eyedrops in acute allergic conjunctivitis] 30 Jan 1997
• Synthesis and identification of the primary degradation product in a commercial ophthalmic formulation using NMR, MS, and a stability-indicating HPLC method for antazoline and naphazoline. 30 Mar 1995
• Evidence for two different imidazoline sites on pancreatic B cells and vascular bed in rat. 22 Feb 1995
• Effects of imidazolines and derivatives on insulin secretion and vascular resistance in perfused rat pancreas. 9 Mar 1994
• Antagonism of levcromakalim by imidazoline- and guanidine-derivatives in rat portal vein: involvement of the delayed rectifier. 29 Nov 1993
• [Nitrosamine formation via non-prescription drugs?] 4 Sep 1993
• [A case of allergic reaction to the sting by the bee] 30 Dec 1992
• Imidazoline antagonists of alpha 2-adrenoceptors increase insulin release in vitro by inhibiting ATP-sensitive K+ channels in pancreatic beta-cells. 30 Aug 1992

See a longer list of these articles.

Technical information about 'Antazoline'

Definition: An antagonist of histamine H1 receptors.

Chemical name: 1H-Imidazole-2-methanamine, 4,5-dihydro-N-phenyl-N-(phenylmethyl)-

Registry Number: 91-75-8

Descriptor UI: D000865

Alternative terms: Antazoline; Phenazoline; Imidamine; Arithmin; Lannett Brand of Antazoline Phosphate; Antazoline Phosphate (1:1); Antasten; Antazoline Hydrochloride; Hydrochloride, Antazoline; Antazoline Phosphate; Phosphate, Antazoline; Antistine; Analergine;

Allowable Qualifiers: administration & dosage; adverse effects; analogs & derivatives; analysis; antagonists & inhibitors; blood; cerebrospinal fluid; chemical synthesis; classification; diagnostic use; economics; history; immunology; isolation & purification; metabolism; pharmacokinetics; pharmacology; poisoning; radiation effects; standards; supply & distribution; therapeutic use; toxicity; urine; chemistry; contraindications; agonists;

Pharmacological Action: Histamine H1 Antagonists; Anti-Allergic Agents;

Tree Number: D03.383.129.308.040;

History Note: 91(75); was see under IMIDAZOLES 1975-90